Bioactive Small Molecules

N'-[1-(4-aminophenyl)ethylidene]-2-iodobenzohydrazide

BLT-5

BLT-5 (click to show)
BLT-5 (click to hide)
Title:
Discovery of chemical inhibitors of the selective transfer of lipids mediated by the HDL receptor SR-BI
Reference:
PNAS November 26, 2002 vol. 99 no. 24 15422-15427
Authors:
Thomas J. F. Nieland, Marsha Penman, Limor Dori, Monty Krieger, and Tomas Kirchhausen
Compounds:
BLT-1 (5234221), BLT-2 (5234225), BLT-3 (5106931), BLT-4 (5109586), BLT-5 (5117098)
BLT-5 (click to show)
BLT-5 (click to hide)
Title:
Identification of the Molecular Target of Small Molecule Inhibitors of HDL Receptor SR-BI Activity
Reference:
Biochemistry, 2008 Jan 8;47(1):460-72. Epub 2007 Dec 8.
Authors:
Thomas J. F. Nieland, Jared T. Shaw, Firoz A. Jaipuri, Jay L. Duffner, Angela N. Koehler, Sotirios Banakos, Vassilis I. Zannis, Tomas Kirchhausen, and Monty Krieger
Compounds:
Compound 1 (5136875), Compound 2 (5136871), Compound 3 (5234224), Compound 4 (5234954), Compound 5 (5554654), Compound 6 (8016115), Compound 7 (8016113), Compound 8 (5153618), Compound 9 (5136957), BLT-1 (5234221), BLT-2 (5234225), BLT-3 (5106931), BLT-4 (5109586), BLT-5 (5117098), BLT-1sc (5152562)