Bioactive Small Molecules

Compound 1, Compound 5, H2L 7905958

H2L 7905958 (click to show)

H2L 7905958 (click to hide)

Title:

Virtual screening approaches for the identification of non-lipid autotaxin inhibitors

Reference:

Bioorg Med Chem. 2008 Feb 15;16(4):1784-95

Authors:

Parrill AL, Echols U, Nguyen T, Pham TC, Hoeglund A, Baker DL

Compounds:

H2L 7905958 (7905958)

Compound 5 (click to show)

Compound 5 (click to hide)

Title:

Characterization of non-lipid autotaxin inhibitors

Reference:

Bioorganic & Medicinal Chemistry, 2010 Jan 15;18(2):769-76. doi: 10.1016/j.bmc.2009.11.056. Epub 2009 Nov 27.

Authors:

Adrienne B. Hoeglund, Angela L. Howard, Irene W. Wanjala, Truc Chi T. Pham, Abby L. Parrill, Daniel L. Baker

Compounds:

Compound 1 (5210574), Compound 2 (5761473), Compound 3 (5564949), Compound 4 (7839888), Compound 5 (7905958), Compound 6 {Not in our database}

Compound 1 (click to show)

Compound 1 (click to hide)

Title:

Optimization of a Pipemidic Acid Autotaxin Inhibitor

Reference:

Journal of Medicinal Chemistry 2010 Feb 11;53(3):1056-66.

Authors:

Adrienne B. Hoeglund, Heidi E. Bostic, Angela L. Howard, Irene W. Wanjala, Michael D. Best, Daniel L. Baker, Abby L. Parrill

Compounds:

Compound 1 (7905958)