Bioactive Small Molecules

3-amino-N-isopropyl-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide

Compound 12

Compound 12 (click to show)
Compound 12 (click to hide)
Title:
An allosteric potentiator of M4 mAChR modulates hippocampal synaptic transmission
Reference:
Nature Chemical Biology 2008 Jan;4(1):42-50.
Authors:
Jana K Shirey, Zixiu Xiang, Darren Orton, Ashley E Brady, Kari A Johnson, Richard Williams, Jennifer E Ayala, Alice L Rodriguez, Jurgen Wess, David Weaver, Colleen M Niswender, & P Jeffrey Conn
Compounds:
Compound 12 (7904200), Compound 15 (7911703), Compound 16 (7912361)