Bioactive Small Molecules

Compound 1

Compound 1 (click to show)

Compound 1 (click to hide)

Title:

Inhibitors of Androgen Receptor Activation Function-2 (AF2) Site Identified through Virtual Screening

Reference:

J Med Chem. 2011 Sep 22;54(18):6197-205. doi: 10.1021/jm200532b. Epub 2011 Aug 29.

Authors:

Peter Axerio-Cilies, Nathan A. Lack, M. Ravi Shashi Nayana, Ka Hong Chan, Anthony Yeung, Eric Leblanc, Emma S. Tomlinson Guns, Paul S. Rennie, and Artem Cherkasov

Compounds:

Compound 4 (5710542), Compound 1 (5722471)