Bioactive Small Molecules

C146

C146 (click to show)

C146 (click to hide)

Title:

Virtual ligand screening of the p300/CBP histone acetyltransferase: identification of a selective small molecule inhibitor

Reference:

Chem Biol. 2010 May 28;17(5):471-82.

Authors:

Bowers EM, Yan G, Mukherjee C, Orry A, Wang L, Holbert MA, Crump NT, Hazzalin CA, Liszczak G, Yuan H, Larocca C, Saldanha SA, Abagyan R, Sun Y, Meyers DJ, Marmorstein R, Mahadevan LC, Alani RM, Cole PA.

Compounds:

C646 (5838646), C146 (5202146), C375 (6643375)