Bioactive Small Molecules

N-(1-{7-[(9-ethyl-9H-carbazol-3-yl)methyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide

VB-018

VB-018 (click to show)
VB-018 (click to hide)
Title:
Identifying GSK-3β kinase inhibitors of Alzheimer's disease: Virtual screening, enzyme, and cell assays
Reference:
Eur J Pharm Sci. 2016 Apr 14;89:11-19. doi: 10.1016/j.ejps.2016.04.012. [Epub ahead of print]
Authors:
Lin CH, Hsieh YS, Wu YR, Hsu CJ, Chen HC, Huang WH, Chang KH, Hsieh-Li HM, Su MT, Sun YC, Lee GC, Lee-Chen GJ
Compounds:
VB-018 (18057186), VB-019 (61140540)