Bioactive Small Molecules

methyl 5-[(1-ethylpropyl)amino]-3-(2-furoylamino)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate

H2-005

H2-005 (click to show)
H2-005 (click to hide)
Title:
Discovery of a novel class of diacylglycerol acyltransferase 2 inhibitors with a 1H-pyrrolo[2,3-b]pyridine core
Reference:
Biol Pharm Bull. 2014;37(10):1655-60. Epub 2014 Aug 7
Authors:
Kim MO, Lee S, Choi K, Lee S, Kim H, Kang H, Choi M, Kwon EB, Kang MJ, Kim S, Lee HJ, Lee HS, Kwak YS, Cho S.
Compounds:
H2-003 (13136439), H2-005 (15078035)